Discovery of thiophen-2-ylmethylene bis-dimedone derivatives as novel WRN inhibitors for treating cancers with microsatellite instability

Hwasun Yang, Miso Kang, Seonyeong Jang, Soo Yeon Baek, Jiwon Kim, Gyeong Un Kim, Dongwoo Kim, Junsu Ha, Jong Seung Kim, Cheulhee Jung, Nam Jung Kim, Sung Yup Cho, Woong Hee Shin, Juyong Lee, Junsu Ko, Ansoo Lee, Gyochang Keum, Sanghee Lee, Taek Kang

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Pharmacology, Toxicology and Pharmaceutical Science

Chemistry